Last Updated on November 26, 2025 by Bilal Hasdemir

Many drugs are used to treat breast cancer. Each drug has its own role and use. For international patients looking for top-notch care, it can be hard to understand all the chemotherapy pill names for breast cancer.
Drugs like tamoxifen, letrozole (Femara), abemaciclib (Verzenio), and trastuzumab (Herceptin) are approved by the FDA. We want to give you a detailed look at these drugs. This way, patients can make better choices about their treatment.
Key Takeaways
- Many drugs are used to treat breast cancer, depending on the stage and type.
- At Liv Hospital, we focus on giving care that uses the newest research and treatments.
- Tamoxifen and letrozole are commonly used hormonal therapies.
- Abemaciclib (Verzenio) is a targeted therapy used in certain cases.
- Trastuzumab (Herceptin) is a monoclonal antibody therapy.
- Understanding treatment options is key to making informed decisions.
Understanding Breast Cancer Medications
Medications are key in treating breast cancer. They come in many types, each suited for different patients. Finding the right one can be tough, but it’s essential for good care.
The Role of Medications in Breast Cancer Treatment
Medications are a big part of breast cancer treatment. They help shrink tumors, kill cancer cells, or stop the cancer from coming back. The right medicine depends on the cancer’s stage, hormone receptors, and the patient’s health.
There are several types of breast cancer medications, including:
- Chemotherapy: Uses drugs to destroy cancer cells.
- Hormone therapy: Works on breast cancers with hormone receptors.
- Targeted therapy: Targets specific characteristics of cancer cells.
The Canadian Cancer Society says targeted therapy uses drugs to target cancer cells’ specific traits.
How Breast Cancer Drugs Are Classified
Breast cancer drugs are sorted by how they work, the cancer type they treat, and how they’re given. Knowing how these drugs are grouped helps patients choose their treatment wisely.
The main groups are:
- Chemotherapy drugs: These are divided into classes based on their action.
- Hormone therapies: These are grouped by whether they block hormone production or affect hormone receptors.
- Targeted therapies: These are sorted by the specific target in the cancer cell.
Comprehensive List of Breast Cancer Drug Names
Understanding breast cancer treatment involves knowing the different medications. There are many breast cancer drug names. Knowing the most common ones can help patients feel more in control of their treatment.
FDA-Approved Medications Overview
The FDA checks breast cancer drugs for safety and effectiveness. FDA-approved breast cancer drugs fall into hormone therapy, chemotherapy, and targeted therapy. We’ll look at these categories to understand breast cancer treatment drugs better.
Some key FDA-approved medications include:
- Anastrozole (Arimidex)
- Exemestane (Aromasin)
- Palbociclib (Ibrance)
- Letrozole (Femara)
These drugs are used at different stages of breast cancer treatment. For more information, visit Cancer Research UK.
Most Commonly Prescribed Options
Some breast cancer drug names are prescribed more often. This is because they are effective and safe. These include:
- Tamoxifen: A hormone therapy for ER-positive breast cancer.
- Trastuzumab (Herceptin): A targeted therapy for HER2-positive breast cancer.
- Cyclophosphamide: A chemotherapy drug used with other treatments.
Knowing about these drugs helps patients understand their treatment plans better.
How to Identify Your Medication
It’s important to know your medication. Here are some tips:
- Always check the name on the packaging.
- Verify dosage instructions with your healthcare provider.
- Know what your medication looks like, including color, shape, and size.
Being informed about your breast cancer treatment drugs helps you work better with your healthcare team.
Hormone Therapy Medications for Breast Cancer
For those with hormone receptor-positive breast cancer, hormone therapy is key. These treatments target cancer cells that estrogen or progesterone fuel.
Tamoxifen: The Pioneering Treatment
Tamoxifen is an anti-estrogen drug used for years to fight hormone receptor-positive breast cancer. It blocks estrogen from reaching cancer cells. Tamoxifen has been shown to significantly reduce the risk of breast cancer recurrence and is given to both pre- and post-menopausal women.
Letrozole (Femara): Aromatase Inhibitor
Letrozole, or Femara, is an aromatase inhibitor. It lowers estrogen levels in the body. By stopping the aromatase enzyme, letrozole slows cancer cell growth. This medication is typically prescribed for post-menopausal women.
Anastrozole (Arimidex): For ER-Positive Disease
Anastrozole, or Arimidex, is another aromatase inhibitor for hormone receptor-positive breast cancer. It works like letrozole by reducing estrogen. Anastrozole is given to post-menopausal women with ER-positive breast cancer.
Exemestane (Aromasin): Post-Menopause Option
Exemestane, or Aromasin, is an aromatase inhibitor for post-menopausal women with hormone receptor-positive breast cancer. It blocks the aromatase enzyme, lowering estrogen levels. This slows cancer cell growth.
These hormone therapy medications offer various treatment options for hormone receptor-positive breast cancer. Understanding these options helps patients make informed decisions with their healthcare providers.
Chemotherapy Pills for Breast Cancer
Chemotherapy pills are a key part of treating breast cancer. They offer a pill form instead of the usual infusion therapy. This makes treatment easier and less scary for many patients.
Capecitabine (Xeloda): Oral Alternative to Infusions
Capecitabine, known as Xeloda, is a pill for breast cancer treatment. The Canadian Cancer Society says it’s used for cancer that has spread. This pill stops cancer cells from growing by messing with their DNA. It’s for patients who haven’t done well with other treatments.
Cyclophosphamide: Traditional Chemotherapy Option
Cyclophosphamide is a long-used chemotherapy drug for breast cancer. It can be given as a pill or through an IV. This flexibility is great for treatments that use different ways to give the drug. It kills cancer cells by damaging their DNA.
Benefits of Oral Chemotherapy Administration
Oral chemotherapy has big benefits for breast cancer patients. It’s easy to take at home, not in a hospital. This makes life easier and less stressful. It also helps the medicine work better over time.
Oral pills also lower the chance of problems from IV treatments. But, patients must take their pills as told and tell their doctor about any side effects.
Targeted Therapy Breast Cancer Pills
Targeted therapy has changed how we treat breast cancer, bringing hope to many. It focuses on cancer cells, not healthy ones. This has led to new drugs that help patients more.
We’ll look at three key pills: palbociclib (Ibrance), abemaciclib (Verzenio), and alpelisib (Piqray). They’ve shown great results in trials and are now part of treatments.
Palbociclib (Ibrance): CDK4/6 Inhibitor
Palbociclib, or Ibrance, is a CDK4/6 inhibitor. It blocks proteins that help cancer cells grow. Studies show it improves survival when used with hormone therapy for certain breast cancers.
Abemaciclib (Verzenio): For Advanced Breast Cancer
Abemaciclib, or Verzenio, is another CDK4/6 inhibitor. It’s special because it can reach brain tumors. It’s used with hormone therapy for advanced breast cancer.
Alpelisib (Piqray): PI3K Inhibitor
Alpelisib, or Piqray, targets a different pathway in cancer cells. It’s used with fulvestrant for certain breast cancers. Its approval was a big step forward for breast cancer treatment.
These pills are big steps forward in breast cancer treatment. Knowing about them helps patients and doctors choose the best treatment.
- Palbociclib (Ibrance): Effective for HR-positive, HER2-negative advanced breast cancer.
- Abemaciclib (Verzenio): Used for HR-positive, HER2-negative advanced or metastatic breast cancer, with the added benefit of crossing the blood-brain barrier.
- Alpelisib (Piqray): Targets PIK3CA-mutated advanced or metastatic breast cancer, providing a new treatment option for patients with specific genetic mutations.
HER2-Targeted Breast Cancer Drugs
HER2-targeted therapies have changed how we treat HER2-positive breast cancer. They target the HER2 protein, found in some cancer cells. This has greatly improved treatment results.
Trastuzumab (Herceptin): Revolutionary HER2 Treatment
Trastuzumab, or Herceptin, was a big step forward in treating HER2-positive breast cancer. It binds to the HER2 protein, slowing cancer cell growth. Studies show it boosts survival rates when paired with chemotherapy.
Trastuzumab brought new hope to those with HER2-positive breast cancer. It marked a major leap in treatment options.
Fam-trastuzumab deruxtecan-nxki (Enhertu): Antibody-Drug Conjugate
Fam-trastuzumab deruxtecan-nxki, or Enhertu, is a new treatment for HER2-positive breast cancer. It combines trastuzumab with a chemotherapy drug, targeting cancer cells directly. Enhertu is approved for those who’ve tried other HER2 treatments, giving them another chance.
Pertuzumab (Perjeta): Combination Therapy Option
Pertuzumab, or Perjeta, is another effective HER2-targeted therapy. It works differently than trastuzumab, adding to its effectiveness. Together with trastuzumab and chemotherapy, pertuzumab boosts survival rates. This combo is now a common treatment for HER2-positive breast cancer.
These therapies have greatly improved treatment for HER2-positive breast cancer. They offer better outcomes and new hope for patients.
Common Medications for Metastatic Breast Cancer
Patients with metastatic breast cancer need to know about their treatment options. This type of cancer has spread to other parts of the body. A treatment plan may include different medications.
Taxanes: Docetaxel and Paclitaxel
Taxanes are a type of chemotherapy used for metastatic breast cancer. Docetaxel and paclitaxel are often prescribed. They help slow down cancer cell growth and spread.
The Canadian Cancer Society says taxanes are very effective. The choice between docetaxel and paclitaxel depends on the patient’s health and past treatments.
| Medication | Common Side Effects | Administration Method |
|---|---|---|
| Docetaxel | Fatigue, hair loss, nausea | Intravenous infusion |
| Paclitaxel | Hair loss, numbness in hands/feet, fatigue | Intravenous infusion |
Eribulin (Halaven): For Late-Stage Treatment
Eribulin, known as Halaven, is used for metastatic breast cancer. It’s for patients who have tried other chemotherapy. Eribulin stops cancer cells from growing.
Studies show eribulin can help patients live longer. Side effects include fatigue, nausea, and hair loss.
Sacituzumab Govitecan (Trodelvy): For Triple-Negative Disease
Sacituzumab govitecan, or Trodelvy, is for triple-negative metastatic breast cancer. It’s for cancers without estrogen or progesterone receptors and too much HER2 protein.
Trodelvy is an antibody-drug conjugate that targets cancer cells. It’s shown to improve survival and slow disease progression in triple-negative cancer.
Knowing about metastatic breast cancer medications is key for patients. They should talk to their healthcare team to find the best treatment plan for them.
Oral vs. Intravenous Breast Cancer Medications
How breast cancer medications are given can change a patient’s treatment and results. We need to look at the differences between oral and intravenous medications. This helps us see how each affects patient care.
Comparing Administration Methods
Oral chemotherapy, like capecitabine (Xeloda), is taken at home. This can cut down on hospital visits. It’s good for those with tight schedules or far from treatment centers.
Oral chemotherapy lets patients control their treatment at home. But, they must follow the dosage and schedule closely. Intravenous chemotherapy is given in a clinic. It’s given right away, but might mean more hospital trips.
Adherence and Quality of Life Considerations
How well patients stick to their treatment is key. Oral meds need strict following, which can be hard. Intravenous meds are given by doctors, so there’s less chance of forgetting.
Quality of life also matters. Oral meds let patients keep up with daily life easily. But, intravenous meds mean more hospital visits. Yet, they offer the comfort of professional care.
When Each Method Is Preferred
Choosing between oral and intravenous meds depends on many things. These include the cancer type and stage, patient preference, and health. Oral meds might suit early-stage cancer or those wanting flexibility. Intravenous meds are often for high-dose or advanced cancer treatments.
The best choice should be made with a doctor’s advice. It’s about what’s best for each patient. Knowing the pros and cons helps support patients in their treatment decisions.
Patient Guide to Taking Breast Cancer Pills
Taking breast cancer pills is a key part of your treatment. We’re here to help you understand how to do it right. It’s important to follow your treatment plan closely. We’ll give you tips on managing your medication, dealing with side effects, and talking to your doctor.
Establishing a Medication Routine
Having a regular routine can help you stick to your medication. Here are some tips:
- Take your pills at the same time every day to make it a habit.
- Use a pill box or calendar to keep track of your doses.
- Set reminders on your phone or ask someone to remind you.
- Keep your pills in a place you can see, like your bathroom or kitchen counter.
By following a routine, you can avoid missing doses and get the most from your treatment.
Tracking and Managing Side Effects
Breast cancer pills can cause side effects, from mild to severe. It’s important to track and manage these effects to keep your quality of life good. Here are some ways to help:
- Keep a journal of your side effects and how bad they are.
- Share your journal with your doctor to adjust your treatment if needed.
- Drink plenty of water and eat well to lessen side effects.
- Try alternative therapies like acupuncture or meditation to help with symptoms.
By actively managing side effects, you can lessen their impact on your life and focus on getting better.
Questions to Ask Your Healthcare Provider
Talking well with your healthcare provider is key for good treatment. Here are some questions to ask:
- What are the most common side effects of my medication, and how can I manage them?
- How will we check how my treatment is working, and what changes might be made?
- Are there any possible problems with my breast cancer medication and other drugs I’m taking?
- What support is there to help me deal with treatment challenges?
By asking the right questions, you can be more involved in your treatment and get the best care.
Recent FDA Approved Breast Cancer Drugs
The fight against breast cancer has seen big changes in recent years. Thanks to the FDA, new treatments have come to light. These new treatments are making life better for those fighting breast cancer.
We’re moving towards treatments that are more precise and tailored to each person. This is a big step forward.
Breakthrough Therapies of the Last Five Years
In the last five years, the FDA has approved several groundbreaking treatments. Palbociclib (Ibrance) and fam-trastuzumab deruxtecan-nxki (Enhertu) are two examples. They’ve shown great results in clinical trials, giving hope to many.
Palbociclib has changed the game for those with hormone receptor-positive, HER2-negative advanced breast cancer. Fam-trastuzumab deruxtecan-nxki has also made a big impact, even for those who’ve tried many treatments before.
Emerging Treatment Paradigms
These new treatments are not just adding options but changing how we treat breast cancer. We’re now combining targeted therapies with immunotherapies and other treatments. This approach aims to get better results.
For example, alpelisib (Piqray) paired with fulvestrant is showing great promise. It’s for those with HR-positive, HER2-negative advanced breast cancer and PIK3CA mutations.
What’s in the Approval Pipeline
The pipeline for new breast cancer treatments is full of hope. We have next-generation CDK4/6 inhibitors, new antibody-drug conjugates, and innovative immunotherapies in late-stage trials. As we learn more about breast cancer, we’ll see even better treatments.
The future of breast cancer treatment is bright. We’re moving towards more precise and personalized care. With new treatments on the way, patients will have better options. This will improve their survival and quality of life.
Conclusion: Navigating Your Breast Cancer Medication Journey
Dealing with breast cancer treatment can be tough. But, with the right info and support, patients can make smart choices about their care. We’ve looked at different breast cancer meds, like hormone therapy, chemotherapy, and targeted therapy.
It’s key to know about the various breast cancer meds for effective treatment. Support and education for patients are very important. They help manage side effects and improve life quality.
New treatments and meds are coming up in breast cancer research. This gives hope for better results. We urge patients to talk closely with their doctors to find the best treatment for them.
With good patient support and education, we can help people be more involved in their breast cancer journey. They can make informed choices and handle treatment with confidence.
FAQ
What are the most common breast cancer drug names?
Common breast cancer drugs include tamoxifen and letrozole (Femara). Anastrozole (Arimidex) and exemestane (Aromasin) are also used. Capecitabine (Xeloda), palbociclib (Ibrance), and trastuzumab (Herceptin) are other examples.
What is hormone therapy for breast cancer?
Hormone therapy blocks hormones from reaching cancer cells. This slows or stops hormone receptor-positive breast cancer growth.
What are chemotherapy pills for breast cancer?
Chemotherapy pills like capecitabine (Xeloda) and cyclophosphamide are oral alternatives. They replace traditional intravenous chemotherapy infusions.
What are targeted therapy breast cancer pills?
Targeted therapy pills include palbociclib (Ibrance), abemaciclib (Verzenio), and alpelisib (Piqray). They target specific proteins or genes in cancer cells.
How do I identify my breast cancer medication?
Check the prescription label or medication packaging to identify your medication. You can also ask your healthcare provider or pharmacist.
What are the benefits of oral chemotherapy administration?
Oral chemotherapy offers flexibility and convenience. It may also have fewer side effects than traditional intravenous chemotherapy.
How do I establish a medication routine for breast cancer treatment?
Take your medication at the same time every day. Use a pill box or reminder. Ask your healthcare provider or pharmacist for guidance.
What are the common side effects of breast cancer medications?
Side effects vary by treatment but may include hot flashes and fatigue. Nausea, hair loss, and mood changes are also common.
How do I track and manage side effects of breast cancer medications?
Keep a symptom journal and report changes to your healthcare provider. Follow their advice on managing side effects.
What questions should I ask my healthcare provider about breast cancer medications?
Ask about the benefits and risks of your medication. Discuss side effects, how to manage them, and any concerns about your treatment.
What are recent FDA-approved breast cancer drugs?
Recent approvals include fam-trastuzumab deruxtecan-nxki (Enhertu) and sacituzumab govitecan (Trodelvy). Alpelisib (Piqray) is another example.
What is the difference between oral and intravenous breast cancer medications?
Oral medications are taken by mouth, while intravenous medications are given through a vein. Each has different benefits and drawbacks.
References
- National Cancer Institute. (n.d.). Drugs for breast cancer. Retrieved from https://www.cancer.gov/about-cancer/treatment/drugs/breast
- National Cancer Institute. (n.d.). Approved targeted therapies drug list. Retrieved from https://www.cancer.gov/about-cancer/treatment/types/targeted-therapies/approved-drug-list
- U.S. Food and Drug Administration. (n.d.). Oncology (cancer / hematologic malignancies) approval notifications. Retrieved from https://www.fda.gov/drugs/resources-information-approved-drugs/oncology-cancerhematologic-malignancies-approval-notifications
- Cancer Research UK. (n.d.). Drugs to treat cancer. Retrieved from https://www.cancerresearchuk.org/about-cancer/treatment/drugs
- BreastCancerTrials. (n.d.). Breast cancer drugs and trials. Retrieved from https://www.breastcancertrials.org/BCTIncludes/Resources/BreastCancerDrugs.html

